From: Structural determinant for inducing RORgamma specific inverse agonism triggered by a synthetic benzoxazinone ligand
ROR
γ
α
β
IC50 (uM)
0.043 (+/− 0.01uM; N = 6)
>10 (N = 2)
>1.2 (N = 2)
Selectivity (X)
-
>235
>28.2